Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04363
Ion Channel
Voltage-gated sodium channel type 1 subunit alpha
Peptide Function
Activator
Gene Name
SCN1A
Activity Data (nM)
IC50
Not available
Ki
Not available
EC50
11.6 nM
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
ECRYLFGGCKTTADCCKHLGCRTDLYYCAWDGTF
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
Hm1b
Peptide Species
Heteroscodra maculata (Togo starburst tarantula) (Togo starburst baboon spider)
Peptide Name
Delta-theraphotoxin-Hm1b
CAS Number
Not available
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−80 mV
Temperature
24 °C
Test Method
Patch-clamping
Test Species
HEK293 cell (Homo sapiens embryonic kidney 293 cell)
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available